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Optimization of brain-penetrant picolinamide derived leucine-rich repeat kinase 2 (LRRK2) inhibitors. Anmol Gulati, Charles S. Yeung, Blair Lapointe, Solomon D. Kattar, Hakan Gunaydin, Jack D. Scott, Kaleen K. Childers, Joey L. Methot, Vladimir Simov, Ravi Kurukulasuriya, Barbara Pio, Greg J. Morriello, Ping Liu, Haiqun Tang, Santhosh Neelamkavil, Harold B. Wood, Vanessa L. Rada, Michael J. Ardolino, Xin Cindy Yan, Rachel Palte, Karin Otte, Robert Faltus, Janice Woodhouse, Laxminarayan G. Hegde, Paul Ciaccio, Ellen C. Minnihan, Erin F. DiMauro, Matthew J. Fell, Peter H. Fuller, J. Michael Ellis
, RSC Med. Chem.
, 2021
, 12
, 1164